AssayIndex
Cross-section

Cagrilintide impurity profile

Every named species the index has reported alongside Cagrilintide, how often, at what level, and what its presence implies about the synthesis or the handling. Reporting threshold is 0.05 % area; anything below it is invisible to this page and is silently added to the main peak.

54 recordsmedian 98.69 %spec 96.5 %
Median total impurities 1.31% n=54
Median largest single 0.65% n=54
Worst single observed 1.32% n=54
Named species observed 5 / 5 n=5
Named speciesΔRT (min)Δ mass (Da)Seen inMedian % areaMax % area
open-chain (reduced disulfide, +2 Da)-1.21+2.01696%0.331.07
disulfide-scrambled isomer+0.48mass-identical96%0.211.32
des-C16 diacid (−254 Da)-3.62-254.22596%0.140.98
deamidated (+1 Da)-0.44+0.98496%0.110.72
cagrilintide dimer (intermolecular disulfide)+3.44+3959.30687%0.091.24

open-chain (reduced disulfide, +2 Da)

Retention offset from the main peak
-1.21 min on RG-2
Mass difference
+2.016 Da
Reported in
52 of 54 records (96 %)
Level when reported
median 0.33 %, max 1.07 %
How it separates
Baseline-resolved on the reference method.

disulfide-scrambled isomer

Retention offset from the main peak
+0.48 min on RG-2
Mass difference
mass-identical — chromatography only
Reported in
52 of 54 records (96 %)
Level when reported
median 0.21 %, max 1.32 %
How it separates
Chromatography only. A gradient long enough to separate it; no mass spectrometer of any resolution will.

des-C16 diacid (−254 Da)

Retention offset from the main peak
-3.62 min on RG-2
Mass difference
-254.225 Da
Reported in
52 of 54 records (96 %)
Level when reported
median 0.14 %, max 0.98 %
How it separates
Baseline-resolved on the reference method.

deamidated (+1 Da)

Retention offset from the main peak
-0.44 min on RG-2
Mass difference
+0.984 Da
Reported in
52 of 54 records (96 %)
Level when reported
median 0.11 %, max 0.72 %
How it separates
Baseline-resolved on the reference method.

cagrilintide dimer (intermolecular disulfide)

Retention offset from the main peak
+3.44 min on RG-2
Mass difference
+3959.306 Da
Reported in
47 of 54 records (87 %)
Level when reported
median 0.09 %, max 1.24 %
How it separates
Baseline-resolved on the reference method.

Degradation pathways

Degradants are a handling finding rather than a synthesis finding. A lot that shipped clean and arrived oxidised tells you about the courier, not the chemist.

  • disulfide scrambling above pH 7.5 — the main stability liability
  • aggregation of the open-chain form, which nucleates fibrils rapidly